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Metiamide
CAS No. 34839-70-8
Metiamide( SK&F 92058 )
Catalog No. M20781 CAS No. 34839-70-8
Metiamide is a histamine H2-receptor antagonist .
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 188 | In Stock |
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| 5MG | 170 | In Stock |
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| 10MG | 282 | In Stock |
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| 25MG | 472 | In Stock |
|
| 50MG | 677 | In Stock |
|
| 100MG | 923 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameMetiamide
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NoteResearch use only, not for human use.
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Brief DescriptionMetiamide is a histamine H2-receptor antagonist .
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DescriptionMetiamide is a histamine H2-receptor antagonist .
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In VitroMetiamide (SK&F 92058) is a competitivewith aldehyde substrates and noncompetitive with the Human E3 Aldehyde Dehydrogenase coenzyme, binding to both the free E3 isozyme and the enzyme·coenzyme binary complex with Ki values of 0.92 μM glycolaldehyde as the varied substrate. Data is got as percentage change in GTPase activity induced by metiamide compared with the GTPase activity stimulated by HA (100 μM).
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In Vivo——
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SynonymsSK&F 92058
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PathwayGPCR/G Protein
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TargetHistamine Receptor
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RecptorH2 receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number34839-70-8
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Formula Weight244.38
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Molecular FormulaC9H16N4S2
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Purity>98% (HPLC)
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SolubilityDMSO:2.4 mg/mL (9.82 mM)
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SMILESCNC(=S)NCCSCc1[nH]cnc1C
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Chemical Name1-methyl-3-(2-(((5-methyl-1H-imidazol-4-yl)methyl)thio)ethyl)thiourea
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Blair E L Grund E R Miller I T et al. Metiamide in the Zollinger-Ellison syndrome[J]. The American Journal of Digestive Diseases 1976 20(12):1123-1130.
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