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DC260126
CAS No. 346692-04-4
DC260126( —— )
Catalog No. M20675 CAS No. 346692-04-4
DC260126 is a small-molecule antagonist of FFA1 (GPR40).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 51 | In Stock |
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| 5MG | 48 | In Stock |
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| 10MG | 63 | In Stock |
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| 25MG | 137 | In Stock |
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| 50MG | 211 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameDC260126
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NoteResearch use only, not for human use.
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Brief DescriptionDC260126 is a small-molecule antagonist of FFA1 (GPR40).
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DescriptionDC260126 is a small-molecule antagonist of FFA1 (GPR40) .
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In VitroDC260126 reduces GTP-loading and ERK1/2 phosphorylation stimulated by linoleic acid in GPR40-CHO cells, suppresses palmitic acid potentiated glucose-stimulated insulin secretion, and negatively regulates GPR40 mRNA expression induced by oleic acid in Min6 cells.
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In Vivo——
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Synonyms——
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PathwayCell Cycle/DNA Damage
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TargetGPR
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RecptorGPR40
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Research Area——
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Indication——
Chemical Information
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CAS Number346692-04-4
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Formula Weight307.38
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Molecular FormulaC16H18FNO2S
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Purity>98% (HPLC)
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SolubilityDMSO:100 mg/mL (325.33 mM)
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SMILESCCCCc1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Peng S Ting W Yuren Z et al. DC260126: A Small-Molecule Antagonist of GPR40 that Protects against Pancreatic β-Cells Dysfunction in db/db Mice[J]. PLoS ONE 2013 8(6):e66744-.
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