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DC260126

CAS No. 346692-04-4

DC260126( —— )

Catalog No. M20675 CAS No. 346692-04-4

DC260126 is a small-molecule antagonist of FFA1 (GPR40).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 51 In Stock
5MG 48 In Stock
10MG 63 In Stock
25MG 137 In Stock
50MG 211 In Stock
100MG Get Quote In Stock
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Biological Information

  • Product Name
    DC260126
  • Note
    Research use only, not for human use.
  • Brief Description
    DC260126 is a small-molecule antagonist of FFA1 (GPR40).
  • Description
    DC260126 is a small-molecule antagonist of FFA1 (GPR40) .
  • In Vitro
    DC260126 reduces GTP-loading and ERK1/2 phosphorylation stimulated by linoleic acid in GPR40-CHO cells, suppresses palmitic acid potentiated glucose-stimulated insulin secretion, and negatively regulates GPR40 mRNA expression induced by oleic acid in Min6 cells.
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    GPR
  • Recptor
    GPR40
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    346692-04-4
  • Formula Weight
    307.38
  • Molecular Formula
    C16H18FNO2S
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:100 mg/mL (325.33 mM)
  • SMILES
    CCCCc1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Peng S Ting W Yuren Z et al. DC260126: A Small-Molecule Antagonist of GPR40 that Protects against Pancreatic β-Cells Dysfunction in db/db Mice[J]. PLoS ONE 2013 8(6):e66744-.
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