Sodium gualenate
CAS No. 6223-35-4
Sodium gualenate( Guaiazulenesulfonate sodium )
Catalog No. M20600 CAS No. 6223-35-4
Sodium gualenate (Guaiazulenesulfonate sodium) a hydrophilic derivative of guaiazulene (GA) is an unstable compound. It has anti-inflammatory and wound-healing effects.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 28 | In Stock |
|
| 100MG | 27 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameSodium gualenate
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NoteResearch use only, not for human use.
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Brief DescriptionSodium gualenate (Guaiazulenesulfonate sodium) a hydrophilic derivative of guaiazulene (GA) is an unstable compound. It has anti-inflammatory and wound-healing effects.
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DescriptionSodium gualenate (Guaiazulenesulfonate sodium) a hydrophilic derivative of guaiazulene (GA) is an unstable compound. It has anti-inflammatory and wound-healing effects. (In Vitro):Sodium gualenate is an unstable compound, which is gradually decomposed in the solid state at room temperature. When heated, Sodium gualenate decomposes almost completely within 1 week. It was found that a kneaded mixture of Sodium gualenate and cornstarch (weight ratio; 1:250) for tableting with water is stable. So, during production, Sodium gualenate could be stabilized using water. Sodium gualenate slightly inhibits the histamine release from rat peritoneal mast cells and strongly inhibits the leukocyte emigration induced by fMLP.(In Vivo):Sodium gualenate has been frequently used for the treatment of human gastritis. Cytoprotection is defined as the main mechanism of Sodium gualenate to protect the mucosa of the stomach and the antipeptic actions in vivo have also been shown.
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In Vitro——
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In Vivo——
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SynonymsGuaiazulenesulfonate sodium
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PathwayOthers
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TargetOther Targets
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RecptorOthers
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Research AreaOthers
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Indicationfolic acid antagonists
Chemical Information
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CAS Number6223-35-4
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Formula Weight300.35
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Molecular FormulaC15H17NaO3S
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Purity>98% (HPLC)
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SolubilityDMSO:30 mg/mL (99.88 mM)
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SMILES[Na+].CC(C)c1ccc(C)c2c(cc(C)c2c1)S([O-])(=O)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Cao T Li Y Yang Z et al. Synthesis and Biological Evaluation of 3 8-dimethyl-5-isopropylazulene Derivatives as Anti-gastric Ulcer Agent[J]. Chemical Biology & Drug Design 2016 88(2):264-271.
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