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Barnidipine
CAS No. 104757-53-1
Barnidipine( Mepirodipine (hydrochloride) | YM-09730-5 )
Catalog No. M20511 CAS No. 104757-53-1
Barnidipine is a dihydropyridine calcium channel blocker that has an IC50 value of 0.35 nM in potassium-induced tonic contraction of pig coronary artery.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 28 | In Stock |
|
| 50MG | 27 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameBarnidipine
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NoteResearch use only, not for human use.
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Brief DescriptionBarnidipine is a dihydropyridine calcium channel blocker that has an IC50 value of 0.35 nM in potassium-induced tonic contraction of pig coronary artery.
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DescriptionBarnidipine is a dihydropyridine calcium channel blocker that has an IC50 value of 0.35 nM in potassium-induced tonic contraction of pig coronary artery.
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In Vitro——
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In Vivo——
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SynonymsMepirodipine (hydrochloride) | YM-09730-5
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PathwayGPCR/G Protein
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TargetCalcium Channel
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RecptorCalcium Channel
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Research Area——
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Indication——
Chemical Information
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CAS Number104757-53-1
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Formula Weight528
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Molecular FormulaC27H30ClN3O6
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Purity>98% (HPLC)
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SolubilityDMSO:250 mg/mL (473.48 mM)
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SMILESCl.COC(=O)C1=C(C)NC(C)=C(C1c1cccc(c1)[N+]([O-])=O)C(=O)O[C@H]1CCN(Cc2ccccc2)C1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Kawashima K Toda H Oohata H et al. Antihypertensive and diuretic effects of YM-09730-5 a new calcium antagonist in stroke-prone spontaneously hypertensive rats[J]. Gen Pharmacol 1991 22(2):263-266.
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