Barnidipine

CAS No. 104757-53-1

Barnidipine( Mepirodipine (hydrochloride) | YM-09730-5 )

Catalog No. M20511 CAS No. 104757-53-1

Barnidipine is a dihydropyridine calcium channel blocker that has an IC50 value of 0.35 nM in potassium-induced tonic contraction of pig coronary artery.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 28 In Stock
50MG 27 In Stock
100MG Get Quote In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Barnidipine
  • Note
    Research use only, not for human use.
  • Brief Description
    Barnidipine is a dihydropyridine calcium channel blocker that has an IC50 value of 0.35 nM in potassium-induced tonic contraction of pig coronary artery.
  • Description
    Barnidipine is a dihydropyridine calcium channel blocker that has an IC50 value of 0.35 nM in potassium-induced tonic contraction of pig coronary artery.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    Mepirodipine (hydrochloride) | YM-09730-5
  • Pathway
    GPCR/G Protein
  • Target
    Calcium Channel
  • Recptor
    Calcium Channel
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    104757-53-1
  • Formula Weight
    528
  • Molecular Formula
    C27H30ClN3O6
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:250 mg/mL (473.48 mM)
  • SMILES
    Cl.COC(=O)C1=C(C)NC(C)=C(C1c1cccc(c1)[N+]([O-])=O)C(=O)O[C@H]1CCN(Cc2ccccc2)C1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Kawashima K Toda H Oohata H et al. Antihypertensive and diuretic effects of YM-09730-5 a new calcium antagonist in stroke-prone spontaneously hypertensive rats[J]. Gen Pharmacol 1991 22(2):263-266.
molnova catalog
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