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PKC-theta inhibitor(b)
CAS No. ——
PKC-theta inhibitor(b)( —— )
Catalog No. M20506 CAS No. ——
PKC-theta inhibitor is a selective PKC-θinhibitor(IC50:12 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 134 | Get Quote |
|
| 5MG | 268 | Get Quote |
|
| 10MG | 431 | Get Quote |
|
| 25MG | 853 | Get Quote |
|
| 100MG | Get Quote | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NamePKC-theta inhibitor(b)
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NoteResearch use only, not for human use.
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Brief DescriptionPKC-theta inhibitor is a selective PKC-θinhibitor(IC50:12 nM).
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DescriptionPKC-theta inhibitor is a selective PKC-θinhibitor(IC50:12 nM).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayAngiogenesis
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TargetPKC
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RecptorPKCθ
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Research Area——
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Indication——
Chemical Information
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CAS Number——
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Formula Weight454.4
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Molecular FormulaC20H25F3N6O3?
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Purity>98% (HPLC)
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SolubilityDMSO:62.5 mg/mL?(137.53 mM)
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SMILESCl.NCC1CCC(CNc2nc(NCc3ccccc3OC(F)(F)F)ncc2[N+]([O-])=O)CC1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Cywin C L Dahmann G Iii A S P et al. Discovery of potent and selective PKC-θ inhibitors[J]. Bioorganic & Medicinal Chemistry Letters 2007 17(1):225-230.
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