PKC-theta inhibitor(b)

CAS No. ——

PKC-theta inhibitor(b)( —— )

Catalog No. M20506 CAS No. ——

PKC-theta inhibitor is a selective PKC-θinhibitor(IC50:12 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 134 Get Quote
5MG 268 Get Quote
10MG 431 Get Quote
25MG 853 Get Quote
100MG Get Quote Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    PKC-theta inhibitor(b)
  • Note
    Research use only, not for human use.
  • Brief Description
    PKC-theta inhibitor is a selective PKC-θinhibitor(IC50:12 nM).
  • Description
    PKC-theta inhibitor is a selective PKC-θinhibitor(IC50:12 nM).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Angiogenesis
  • Target
    PKC
  • Recptor
    PKCθ
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    ——
  • Formula Weight
    454.4
  • Molecular Formula
    C20H25F3N6O3?
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:62.5 mg/mL?(137.53 mM)
  • SMILES
    Cl.NCC1CCC(CNc2nc(NCc3ccccc3OC(F)(F)F)ncc2[N+]([O-])=O)CC1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Cywin C L Dahmann G Iii A S P et al. Discovery of potent and selective PKC-θ inhibitors[J]. Bioorganic & Medicinal Chemistry Letters 2007 17(1):225-230.
molnova catalog
related products
  • Indolactam V

    Indolactam V ((-)-Indolactam V) is an indole alkaloid tumor promoter that activates protein kinase C (PKC).

  • Bryostatin 1

    Bryostatin 1 (NSC 339555) is a macrocyclic lactone derived from a marine invertebrate, fuctions as an activator of PKC with high binding affinity (Ki=1.35 nM).

  • Pim-1 kinase inhibit...

    Pim-1 kinase inhibitor 8 is a potent Pim-1 kinase inhibitor with anticancer activity and can effectively inhibit cell migration.