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PKC-theta inhibitor

CAS No. 736048-65-0

PKC-theta inhibitor( —— )

Catalog No. M20187 CAS No. 736048-65-0

PKC-theta inhibitor is PKC-θinhibitor with an IC50 of 12 nM.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
1 mL x 10 mM in DMSO	274	In Stock
5MG	250	In Stock
10MG	330	In Stock
25MG	467	In Stock
50MG	600	In Stock
100MG	923	In Stock
200MG	1237	In Stock
500MG	Get Quote	In Stock
1G	Get Quote	In Stock

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Biological Information

Product Name

PKC-theta inhibitor
Note

Research use only, not for human use.
Brief Description

PKC-theta inhibitor is PKC-θinhibitor with an IC50 of 12 nM.
Description

PKC-theta inhibitor is PKC-θinhibitor with an IC50 of 12 nM.
In Vitro

——
In Vivo

——
Synonyms

——
Pathway

Angiogenesis
Target

PKC
Recptor

PKCθ
Research Area

——
Indication

——

Chemical Information

CAS Number

736048-65-0
Formula Weight

454.4
Molecular Formula

C20H25F3N6O3
Purity

>98% (HPLC)
Solubility

DMSO:62.5 mg/mL?(137.53 mM)
SMILES

NCC1CCC(CNc2nc(NCc3ccccc3OC(F)(F)F)ncc2[N+]([O-])=O)CC1
Chemical Name

N4-((4-(aminomethyl)cyclohexyl)methyl)-5-nitro-N2-(2-(trifluoromethoxy)benzyl)pyrimidine-24-diamine

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Cywin CL et al. Discovery of potent and selective PKC-theta inhibitors. Bioorg Med Chem Lett. 2007 Jan 1;17(1):225-30.

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