Afloqualone

CAS No. 56287-74-2

Afloqualone( HQ-495 )

Catalog No. M19814 CAS No. 56287-74-2

Afloqualone is a agonist of GABA receptor . Target: GABA Receptor in vitro: Afloqualone is a quinazolinone family GABAergic drug. Afloqualone is an analogue of methaqualone.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 57 In Stock
25MG 29 In Stock
50MG 38 In Stock
100MG 52 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Afloqualone
  • Note
    Research use only, not for human use.
  • Brief Description
    Afloqualone is a agonist of GABA receptor . Target: GABA Receptor in vitro: Afloqualone is a quinazolinone family GABAergic drug. Afloqualone is an analogue of methaqualone.
  • Description
    Afloqualone is a agonist of GABA receptor . Target: GABA Receptor in vitro: Afloqualone is a quinazolinone family GABAergic drug. Afloqualone is an analogue of methaqualone. It has sedative and muscle-relaxant effects resulting from its agonist activity at the β subtype of the GABAa receptor.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    HQ-495
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    GABAR
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    56287-74-2
  • Formula Weight
    283.3
  • Molecular Formula
    C16H14FN3O
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:≥33 mg/mL (116.48 mM)
  • SMILES
    Cc1ccccc1-n1c(CF)nc2ccc(N)cc2c1=O
  • Chemical Name
    6-amino-2-(fluoromethyl)-3-(2-methylphenyl)-4(3H)-quinazolinone

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Yamamura M et al. Effects of afloqualone a new centrally acting muscle relaxant on DRL response and CER in rats (author's transl). Nihon Yakurigaku Zasshi. 1981 Oct;78(4):381-92.
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