PRX-08066 Maleic acid

CAS No. 866206-55-5

PRX-08066 Maleic acid( PRX-08066 Maleate )

Catalog No. M19194 CAS No. 866206-55-5

PRX-08066 Maleic acid is a selective 5-HT2B receptor antagonist with IC50 of 3.4 nM, prevents the severity of pulmonary arterial hypertension in the MCT rat model. Phase 2.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 402 In Stock
5MG 171 In Stock
10MG 233 In Stock
25MG 420 In Stock
50MG 606 In Stock
100MG 863 In Stock
200MG 1172 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    PRX-08066 Maleic acid
  • Note
    Research use only, not for human use.
  • Brief Description
    PRX-08066 Maleic acid is a selective 5-HT2B receptor antagonist with IC50 of 3.4 nM, prevents the severity of pulmonary arterial hypertension in the MCT rat model. Phase 2.
  • Description
    PRX-08066 Maleate is a novel potent and selective 5-HT2B receptor antagonist.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    PRX-08066 Maleate
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    5-HT2B
  • Research Area
    Cardiovascular Disease
  • Indication
    ——

Chemical Information

  • CAS Number
    866206-55-5
  • Formula Weight
    517.96
  • Molecular Formula
    C19H17ClFN5S·C4H4O4
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    C1CN(CCC1NC2=C3C=C(SC3=NC=N2)Cl)CC4=CC(=C(C=C4)F)C#N.C(=C\C(=O)O)\C(=O)O
  • Chemical Name
    5-[[4-[(6-Chlorothieno[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl]methyl]-2-fluorobenzonitrile maleate

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

molnova catalog
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