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GSK2830371
CAS No. 1404456-53-6
GSK2830371( GSK 2830371 | GSK2830371 | GSK-2830371 )
Catalog No. M17279 CAS No. 1404456-53-6
GSK2830371 is an orally active, allosteric Wip1 phosphatase inhibitor with IC50 of 6 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 46 | In Stock |
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| 5MG | 46 | In Stock |
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| 10MG | 78 | In Stock |
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| 25MG | 145 | In Stock |
|
| 50MG | 248 | In Stock |
|
| 100MG | 416 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameGSK2830371
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NoteResearch use only, not for human use.
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Brief DescriptionGSK2830371 is an orally active, allosteric Wip1 phosphatase inhibitor with IC50 of 6 nM.
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DescriptionGSK 2830371 is a WiP1 inhibitor. It inhibits cell growth and tumor growth in lymphoma and neuroblastoma models.
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In Vitro——
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In Vivo——
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SynonymsGSK 2830371 | GSK2830371 | GSK-2830371
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PathwayAngiogenesis
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TargetFGFR
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RecptorWip1 phosphatase
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number1404456-53-6
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Formula Weight461.02
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Molecular FormulaC23H29ClN4O2S
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Purity>98% (HPLC)
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SolubilityDMSO : ≥ 51 mg/mL. 110.62 mM
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SMILESCC1=NC=C(Cl)C=C1NCC1=CC=C(S1)C(=O)N[C@@H](CC1CCCC1)C(=O)NC1CC1
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Chemical Name(S)-5-(((5-chloro-2-methylpyridin-3-yl)amino)methyl)-N-(3-cyclopentyl-1-(cyclopropylamino)-1-oxopropan-2-yl)thiophene-2-carboxamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Gilmartin AG, et al. Nat Chem Biol. 2014, 10(3), 181-187
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