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Desmethyl-VS-5584
CAS No. 1246535-95-4
Desmethyl-VS-5584( Desmethyl-VS-5584 | Desmethyl-VS5584 )
Catalog No. M17217 CAS No. 1246535-95-4
Desmethyl-VS-5584 is a dimethyl analog of VS-5584, which is a novel and highly selective PI3K/mTOR kinase inhibitor for the treatment of cancer.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 86 | In Stock |
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| 5MG | 138 | In Stock |
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| 10MG | 243 | In Stock |
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| 25MG | 408 | In Stock |
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| 50MG | 601 | In Stock |
|
| 100MG | 854 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameDesmethyl-VS-5584
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NoteResearch use only, not for human use.
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Brief DescriptionDesmethyl-VS-5584 is a dimethyl analog of VS-5584, which is a novel and highly selective PI3K/mTOR kinase inhibitor for the treatment of cancer.
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DescriptionDesmethyl-VS-5584 is a demethyl analogue of VS-5584, which is a novel and highly selective PI3K/mTOR kinase inhibitor for the treatment of cancer.
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In Vitro——
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In Vivo——
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SynonymsDesmethyl-VS-5584 | Desmethyl-VS5584
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PathwayCell Cycle/DNA Damage
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TargetPARP
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RecptormTOR| PI3K
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Research Area——
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Indication——
Chemical Information
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CAS Number1246535-95-4
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Formula Weight340.39
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Molecular FormulaC16H20N8O
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Purity>98% (HPLC)
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Solubility——
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SMILESNc1ncc(c2c3ncn(C(C)C)c3nc(N3CCOCC3)n2)cn1
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Chemical Name5-[9-(1-Methylethyl)-2-(4-morpholinyl)-9H-purin-6-yl]-2-pyrimidinamine
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Shao Z,et al. VS-5584, a Novel PI3K-mTOR Dual Inhibitor, Inhibits Melanoma Cell Growth In Vitro and In Vivo. PLoS One. 2015 Jul 23;10(7).
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