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CX 04328
CAS No. 957890-42-5
CX 04328( LEDGIN-6 )
Catalog No. M16841 CAS No. 957890-42-5
CX 04328 (LEDGIN-6) is an allosteric HIV-1 integrase inhibitor that inhibits the LEDGF/p75-integrase interaction with IC50 of 1.37 uM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 262 | In Stock |
|
| 50MG | 1188 | In Stock |
|
| 100MG | 1791 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
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Biological Information
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Product NameCX 04328
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NoteResearch use only, not for human use.
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Brief DescriptionCX 04328 (LEDGIN-6) is an allosteric HIV-1 integrase inhibitor that inhibits the LEDGF/p75-integrase interaction with IC50 of 1.37 uM.
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DescriptionCX 04328 (LEDGIN-6) is an allosteric HIV-1 integrase inhibitor that inhibits the LEDGF/p75-integrase interaction with IC50 of 1.37 uM, antiviral activity EC50 of 2.35 uM.
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In Vitro——
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In Vivo——
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SynonymsLEDGIN-6
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PathwayMicrobiology/Virology
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TargetHIV
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RecptorHIV
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Research AreaInfection
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Indication——
Chemical Information
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CAS Number957890-42-5
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Formula Weight353.846
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Molecular FormulaC21H20ClNO2
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Purity>98% (HPLC)
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SolubilityDMSO : ≥ 100 mg/mL 282.61 mM; H2O : < 0.1 mg/mL
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SMILESCCCC(C1=C(C2=CC=CC=C2)C3=CC(Cl)=CC=C3N=C1C)C(O)=O
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Chemical Name2-(6-chloro-2-methyl-4-phenylquinolin-3-yl)pentanoic acid
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Christ F, et al. Nat Chem Biol. 2010 Jun;6(6):442-8.
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