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Home - Products - GPCR/G Protein - Histamine Receptor - MK-7288

MK-7288

CAS No. 936626-07-2

MK-7288( MK7288 | MK 7288 )

Catalog No. M16708 CAS No. 936626-07-2

A novel histamine H3 receptor inverse agonist for the treatment of sleep apnoea syndrome.

Purity : >98% (HPLC)

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Biological Information

  • Product Name
    MK-7288
  • Note
    Research use only, not for human use.
  • Brief Description
    A novel histamine H3 receptor inverse agonist for the treatment of sleep apnoea syndrome.
  • Description
    A novel histamine H3 receptor inverse agonist for the treatment of sleep apnoea syndrome; significantly prolongs MWT sleep latency, and improves car driving simulation standard deviation of lane position in clinical trials.Sleep Disorder Phase 1 Clinical.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    MK7288 | MK 7288
  • Pathway
    GPCR/G Protein
  • Target
    Histamine Receptor
  • Recptor
    Histamine Receptor
  • Research Area
    Neurological Disease
  • Indication
    Sleep Disorder

Chemical Information

  • CAS Number
    936626-07-2
  • Formula Weight
    401.507
  • Molecular Formula
    C22H31N3O4
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CN(CCN1CCCCC1)C(=O)C2CCC3(CC2)C4=C(C(=O)O3)N=C(C=C4)OC
  • Chemical Name
    (1r,4r)-2'-methoxy-N-methyl-7'-oxo-N-(2-(piperidin-1-yl)ethyl)-7'H-spiro[cyclohexane-1,5'-furo[3,4-b]pyridine]-4-carboxamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Sun H, et al. J Clin Pharmacol. 2013 Dec;53(12):1294-302.
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