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MK-7288
CAS No. 936626-07-2
MK-7288( MK7288 | MK 7288 )
Catalog No. M16708 CAS No. 936626-07-2
A novel histamine H3 receptor inverse agonist for the treatment of sleep apnoea syndrome.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 873 | Get Quote |
|
| 50MG | 1782 | Get Quote |
|
| 100MG | 2250 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NameMK-7288
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NoteResearch use only, not for human use.
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Brief DescriptionA novel histamine H3 receptor inverse agonist for the treatment of sleep apnoea syndrome.
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DescriptionA novel histamine H3 receptor inverse agonist for the treatment of sleep apnoea syndrome; significantly prolongs MWT sleep latency, and improves car driving simulation standard deviation of lane position in clinical trials.Sleep Disorder Phase 1 Clinical.
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In Vitro——
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In Vivo——
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SynonymsMK7288 | MK 7288
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PathwayGPCR/G Protein
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TargetHistamine Receptor
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RecptorHistamine Receptor
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Research AreaNeurological Disease
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IndicationSleep Disorder
Chemical Information
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CAS Number936626-07-2
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Formula Weight401.507
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Molecular FormulaC22H31N3O4
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Purity>98% (HPLC)
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Solubility——
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SMILESCN(CCN1CCCCC1)C(=O)C2CCC3(CC2)C4=C(C(=O)O3)N=C(C=C4)OC
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Chemical Name(1r,4r)-2'-methoxy-N-methyl-7'-oxo-N-(2-(piperidin-1-yl)ethyl)-7'H-spiro[cyclohexane-1,5'-furo[3,4-b]pyridine]-4-carboxamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Sun H, et al. J Clin Pharmacol. 2013 Dec;53(12):1294-302.
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