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Lorediplon
CAS No. 917393-39-6
Lorediplon( GF-015535-00 )
Catalog No. M16588 CAS No. 917393-39-6
A partial positive allosteric GABAA receptor modulator.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 41 | In Stock |
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| 10MG | 37 | In Stock |
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| 25MG | 76 | In Stock |
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| 50MG | 144 | In Stock |
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| 100MG | 226 | In Stock |
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| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameLorediplon
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NoteResearch use only, not for human use.
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Brief DescriptionA partial positive allosteric GABAA receptor modulator.
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DescriptionA partial positive allosteric GABAA receptor modulator; displays activity at the alpha1-subunit, associated with promoting sleep.Sleep Disorder Phase 1 Clinical.
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In Vitro——
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In Vivo——
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SynonymsGF-015535-00
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PathwayMembrane Transporter/Ion Channel
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TargetGAT
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RecptorGAT
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Research AreaNeurological Disease
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IndicationSleep Disorder
Chemical Information
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CAS Number917393-39-6
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Formula Weight394.4221
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Molecular FormulaC20H15FN4O2S
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Purity>98% (HPLC)
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Solubility10 mM in DMSO
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SMILESCC(N(C1=CC(C2=CC=NC3=C(C(C4=CC=CS4)=O)C=NN23)=CC=C1F)C)=O
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Chemical NameAcetamide, N-[2-fluoro-5-[3-(2-thienylcarbonyl)pyrazolo[1,5-a]pyrimidin-7-yl]phenyl]-N-methyl-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Zisapel N. Expert Opin Investig Drugs. 2015 Mar;24(3):401-11.
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