Cart
sales@molnova.com
Lorediplon
CAS No. 917393-39-6
Lorediplon( GF-015535-00 )
Catalog No. M16588 CAS No. 917393-39-6
A partial positive allosteric GABAA receptor modulator.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 10MG | 35 | Get Quote |
|
| 25MG | 72 | Get Quote |
|
| 50MG | 140 | Get Quote |
|
| 100MG | 219 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
-
Product NameLorediplon
-
NoteResearch use only, not for human use.
-
Brief DescriptionA partial positive allosteric GABAA receptor modulator.
-
DescriptionA partial positive allosteric GABAA receptor modulator; displays activity at the alpha1-subunit, associated with promoting sleep.Sleep Disorder Phase 1 Clinical.
-
In Vitro——
-
In Vivo——
-
SynonymsGF-015535-00
-
PathwayMembrane Transporter/Ion Channel
-
TargetGAT
-
RecptorGAT
-
Research AreaNeurological Disease
-
IndicationSleep Disorder
Chemical Information
-
CAS Number917393-39-6
-
Formula Weight394.4221
-
Molecular FormulaC20H15FN4O2S
-
Purity>98% (HPLC)
-
Solubility10 mM in DMSO
-
SMILESCC(N(C1=CC(C2=CC=NC3=C(C(C4=CC=CS4)=O)C=NN23)=CC=C1F)C)=O
-
Chemical NameAcetamide, N-[2-fluoro-5-[3-(2-thienylcarbonyl)pyrazolo[1,5-a]pyrimidin-7-yl]phenyl]-N-methyl-
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Zisapel N. Expert Opin Investig Drugs. 2015 Mar;24(3):401-11.
molnova catalog
related products
-
GR3027
GR3027 (Golexanolone) is a GABA-A receptor modulating steroid antagonist that selectively antagonizes the enhanced activation of GABAA receptors by neurosteroids such as allopregnanolone and THDOC.
-
HZ-166
HZ-166 (HZ166) is a GABAA receptor subtype-selective benzodiazepine site ligand with preferential activity at α2- and α3-GABA(A) receptors.
-
Lesogaberan
Lesogaberan (AZD-3355) is a potent, selective, peripherally acting GABAB receptor agonist with Ki of 5 nM and EC50 of 8.6 nM, 274-fold selectivity over GABAA (Ki=1.4 uM).
