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TAK-100
CAS No. 907609-33-0
TAK-100( TAK100 )
Catalog No. M16521 CAS No. 907609-33-0
TAK-100 is a potent, selective and orally active inhibitor of DPP-4 with IC50 of 5.3 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 100MG | Get Quote | Get Quote |
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| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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| 100MG | Get Quote | Get Quote |
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| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NameTAK-100
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NoteResearch use only, not for human use.
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Brief DescriptionTAK-100 is a potent, selective and orally active inhibitor of DPP-4 with IC50 of 5.3 nM.
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DescriptionTAK-100 is a potent, selective and orally active inhibitor of DPP-4 with IC50 of 5.3 nM, shows no inhibition on DPP2/8/9.Diabetes Phase 1 Discontinued.
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In Vitro——
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In Vivo——
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SynonymsTAK100
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PathwayMetabolic Enzyme/Protease
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TargetDPP
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RecptorDPP
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Research AreaMetabolic Disease
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IndicationDiabetes
Chemical Information
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CAS Number907609-33-0
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Formula Weight354.494
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Molecular FormulaC22H30N2O2
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical Name[5-(aminomethyl)-6-(2,2-dimethylpropyl)-2-ethyl4-(4-methylphenyl)pyridin-3-yl]acetic acid
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Miyamoto Y, et al. J Med Chem. 2011 Feb 10;54(3):831-50.
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