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CeMMEC2
CAS No. 902955-25-3
CeMMEC2( CeMMEC 2 )
Catalog No. M16491 CAS No. 902955-25-3
CeMMEC2 is a novel potent BRD4 inhibitor with IC50 of 0.9 uM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 873 | Get Quote |
|
| 50MG | 1782 | Get Quote |
|
| 100MG | 2250 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NameCeMMEC2
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NoteResearch use only, not for human use.
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Brief DescriptionCeMMEC2 is a novel potent BRD4 inhibitor with IC50 of 0.9 uM.
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DescriptionCeMMEC2 is a novel potent BRD4 inhibitor with IC50 of 0.9 uM, binds to both bromodomains of BRD4, comparably to (S)-JQ1.
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In Vitro——
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In Vivo——
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SynonymsCeMMEC 2
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PathwayChromatin/Epigenetic
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TargetBromodomain
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RecptorBromodomain
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Research Area——
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Indication——
Chemical Information
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CAS Number902955-25-3
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Formula Weight257.34
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Molecular FormulaC14H19N5
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Purity>98% (HPLC)
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Solubility——
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SMILESCC1=NN=C2C=CC(NCCC3=CCCCC3)=NN21
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Chemical NameN-[2-(cyclohex-1-en-1-yl)ethyl]-3-methyl[1,2,4]triazolo[4,3-b]pyridazin-6-amine
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Sdelci S, et al. Nat Chem Biol. 2016 Jul;12(7):504-10.
2. Blank, J. et al. WPO patent WO/2014/191894 (2014).
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