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WDR5-0103
CAS No. 890190-22-4
WDR5-0103( WD-Repeat Protein 5-0103 )
Catalog No. M16426 CAS No. 890190-22-4
A potent MLL1-WDR5 interaction inhibitor with IC50 of 26.4 nM in competitive binding assay.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 35 | In Stock |
|
| 5MG | 57 | In Stock |
|
| 10MG | 96 | In Stock |
|
| 25MG | 197 | In Stock |
|
| 50MG | 347 | In Stock |
|
| 100MG | 516 | In Stock |
|
| 500MG | 1125 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameWDR5-0103
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NoteResearch use only, not for human use.
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Brief DescriptionA potent MLL1-WDR5 interaction inhibitor with IC50 of 26.4 nM in competitive binding assay.
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DescriptionA potent MLL1-WDR5 interaction inhibitor with IC50 of 26.4 nM in competitive binding assay; inhibits the catalytic activity of MLL1 complex with IC50 value of 5.4 uM.
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In Vitro——
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In Vivo——
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SynonymsWD-Repeat Protein 5-0103
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PathwayChromatin/Epigenetic
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TargetHMTase
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RecptorWDR5
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number890190-22-4
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Formula Weight383.4409
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Molecular FormulaC21H25N3O4
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Purity>98% (HPLC)
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SolubilityDMSO: ≥ 40 mg/mL
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SMILESO=C(OC)C1=CC(NC(C2=CC=CC(OC)=C2)=O)=C(N3CCN(C)CC3)C=C1
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Chemical NameBenzoic acid, 3-[(3-methoxybenzoyl)amino]-4-(4-methyl-1-piperazinyl)-, methyl ester
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Li DD, et al. Bioorg Med Chem. 2016 Nov 15;24(22):6109-6118.
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