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AKT Kinase Inhibitor
CAS No. 842148-40-7
AKT Kinase Inhibitor( —— )
Catalog No. M16130 CAS No. 842148-40-7
An Akt kinase inhibitor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 312 | In Stock |
|
| 10MG | 537 | In Stock |
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| 25MG | 842 | In Stock |
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| 50MG | 1134 | In Stock |
|
| 100MG | 1521 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
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Biological Information
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Product NameAKT Kinase Inhibitor
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NoteResearch use only, not for human use.
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Brief DescriptionAn Akt kinase inhibitor.
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DescriptionAn Akt kinase inhibitor.
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In VitroThe effect of selective inhibition of Akt in proliferating cells expressing Trop-2 is studied.Akt inhibition, either by silencing or with specific drugs, induces a marked decrease in cell proliferation in cells expressing Trop-2, in a dose-dependent fashion.
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In VivoTrop-2 expressing tumors subcutaneously injected in animal models show a striking reduction of growth following treatment with specific drugs that inhibit Akt activity. Therefore Akt has a central functional role in mediating the Trop-2-dependent growth stimulus.
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Synonyms——
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PathwayCytoskeleton/Cell Adhesion Molecules
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TargetAkt
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RecptorAkt
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number842148-40-7
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Formula Weight357.3672
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Molecular FormulaC16H19N7O3
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Purity>98% (HPLC)
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Solubility10 mM in DMSO
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SMILESCCN1C2=C(C(=NC=C2OCCCN)C#CCO)N=C1C3=NON=C3N
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Chemical Name2-Propyn-1-ol, 3-[2-(4-amino-1,2,5-oxadiazol-3-yl)-7-(3-aminopropoxy)-1-ethyl-1H-imidazo[4,5-c]pyridin-4-yl]-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
molnova catalog
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