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WH-4-023
CAS No. 837422-57-8
WH-4-023( WH-4-023 | WH4-023 | WH 4-023 | WH-4023 )
Catalog No. M16103 CAS No. 837422-57-8
WH-4-023 is a potent and orally active Lck/Src inhibitor with IC50 of 2 nM and 6 nM in cell-free assays, respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 42 | In Stock |
|
| 5MG | 61 | In Stock |
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| 10MG | 91 | In Stock |
|
| 25MG | 149 | In Stock |
|
| 50MG | 186 | In Stock |
|
| 100MG | 332 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameWH-4-023
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NoteResearch use only, not for human use.
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Brief DescriptionWH-4-023 is a potent and orally active Lck/Src inhibitor with IC50 of 2 nM and 6 nM in cell-free assays, respectively.
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DescriptionWH-4-023 is a potent and orally active Lck/Src inhibitor with IC50 of 2 nM and 6 nM in cell-free assays, respectively.
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In Vitro——
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In Vivo——
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SynonymsWH-4-023 | WH4-023 | WH 4-023 | WH-4023
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PathwayTyrosine Kinase
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TargetSrc
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RecptorLck| Src
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number837422-57-8
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Formula Weight568.67
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Molecular FormulaC32H36N6O4
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Purity>98% (HPLC)
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SolubilityEthanol: 6 mg/mL warmed (10.55 mM); DMSO: 12 mg/mL warmed (21.1 mM)
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SMILESO=C(OC1=C(C)C=CC=C1C)N(C2=CC=C(OC)C=C2OC)C3=NC(NC4=CC=C(N5CCN(C)CC5)C=C4)=NC=C3
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Chemical Name2,6-dimethylphenyl (2,4-dimethoxyphenyl)(2-((4-(4-methylpiperazin-1-yl)phenyl)amino)pyrimidin-4-yl)carbamate
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Martin MW, et al. J Med Chem. 2006 Aug 10;49(16): 4981-9
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