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Elvitegravir
CAS No. 697761-98-1
Elvitegravir( GS-9137, JTK-303 )
Catalog No. M15676 CAS No. 697761-98-1
Elvitegravir (GS-9137, JTK-303) is an HIV integrase inhibitor for HIV-1 IIIB, HIV-2 EHO and HIV-2 ROD with IC50 of 0.7 nM, 2.8 nM and 1.4 nM in cell-free assays, respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 45 | In Stock |
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| 5MG | 45 | In Stock |
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| 10MG | 75 | In Stock |
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| 25MG | 147 | In Stock |
|
| 50MG | 277 | In Stock |
|
| 100MG | 452 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameElvitegravir
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NoteResearch use only, not for human use.
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Brief DescriptionElvitegravir (GS-9137, JTK-303) is an HIV integrase inhibitor for HIV-1 IIIB, HIV-2 EHO and HIV-2 ROD with IC50 of 0.7 nM, 2.8 nM and 1.4 nM in cell-free assays, respectively.
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DescriptionElvitegravir (GS-9137, JTK-303) is an HIV integrase inhibitor for HIV-1 IIIB, HIV-2 EHO and HIV-2 ROD with IC50 of 0.7 nM, 2.8 nM and 1.4 nM in cell-free assays, respectively.
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In Vitro——
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In Vivo——
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SynonymsGS-9137, JTK-303
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PathwayMicrobiology/Virology
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TargetHIV
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RecptorHIV-1 IIIB| HIV-2 EHO| HIV-2 ROD
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Research AreaInfection
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Indication——
Chemical Information
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CAS Number697761-98-1
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Formula Weight447.88
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Molecular FormulaC23H23ClFNO5
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Purity>98% (HPLC)
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SolubilityEthanol: 35 mg/mL (78.14 mM); DMSO: 90 mg/mL (200.94 mM)
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SMILESCC(C)[C@@H](CO)N1C=C(C(=O)C2=CC(=C(C=C21)OC)CC3=C(C(=CC=C3)Cl)F)C(=O)O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Shimura K, et al. J Virol. 2008, 82(2), 764-774.
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