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CP-724714 (b)
CAS No. 537705-08-1
CP-724714 (b)( —— )
Catalog No. M14915 CAS No. 537705-08-1
CP-724714 is a potent, selective inhibitor of HER2/ErbB2 with IC50 of 10 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 873 | In Stock |
|
| 50MG | 1782 | In Stock |
|
| 100MG | 2250 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameCP-724714 (b)
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NoteResearch use only, not for human use.
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Brief DescriptionCP-724714 is a potent, selective inhibitor of HER2/ErbB2 with IC50 of 10 nM.
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DescriptionCP-724714 is a potent, selective inhibitor of HER2/ErbB2 with IC50 of 10 nM, >640-fold selectivity against EGFR, InsR, IRG-1R, PDGFR, VEGFR2, Abl, Src, c-Met etc in cell-free assays. Phase 2.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayAngiogenesis
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TargetEGFR
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RecptorHER2/ErbB2
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number537705-08-1
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Formula Weight469.53
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Molecular FormulaC27H27N5O3
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Purity>98% (HPLC)
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SolubilityN/A
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SMILESCCOC(=O)NC/C=C/C1=CC2=C(C=C1)N=CN=C2NC3=CC(=C(C=C3)OC4=CN=C(C=C4)C)C
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1 Jani JP, et al. Cancer Res, 2007, 67(20), 9887-9893.
2 Feng B, et al. Toxicol Sci, 2009, 108(2), 492-500.
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