Enoxolone
CAS No. 471-53-4
Enoxolone( Arthrodont | Biosone | Enoxolone | α-Glycyrrhetinic Acid? | GM 1658 | NSC 35347 | PO 12 | STX 352 )
Catalog No. M14567 CAS No. 471-53-4
Enoximone is a selective phosphodiesterase inhibitor with vasodilating and positive inotropic activity that does not cause changes in myocardial oxygen consumption.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 500MG | 39 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameEnoxolone
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NoteResearch use only, not for human use.
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Brief DescriptionEnoximone is a selective phosphodiesterase inhibitor with vasodilating and positive inotropic activity that does not cause changes in myocardial oxygen consumption.
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DescriptionEnoximone is a selective phosphodiesterase inhibitor with vasodilating and positive inotropic activity that does not cause changes in myocardial oxygen consumption. It is used in patients with congestive heart failure. Trials were halted in the U.S., but the drug is used in various countries.
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In Vitro——
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In Vivo——
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SynonymsArthrodont | Biosone | Enoxolone | α-Glycyrrhetinic Acid? | GM 1658 | NSC 35347 | PO 12 | STX 352
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PathwayMetabolic Enzyme/Protease
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TargetDehydrogenase
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RecptorDHO
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Research AreaOther Indications
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Indication——
Chemical Information
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CAS Number471-53-4
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Formula Weight470.68
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Molecular FormulaC30H46O4
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Purity>98% (HPLC)
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SolubilityDMSO: 94 mg/mL (199.71 mM)
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SMILESCC(C)([C@](CC[C@@]([C@@]1(CC[C@]2(CC[C@](C(O)=O)(C[C@]2(C1=C3)[H])C)C)C)4C)5[H])[C@@H](O)CC[C@]5(C)[C@@]4([H])C3=O
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Chemical Name(2S,4aS,6aS,6bR,8aR,10S,12aS,12bR,14bR)-10-hydroxy-2,4a,6a,6b,9,9,12a-heptamethyl-13-oxo-1,2,3,4,4a,5,6,6a,6b,7,8,8a,9,10,11,12,12a,12b,13,14b-icosahydropicene-2-carboxylic acid
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Boldt J, et al. Expert Opin PharmacOthers. 2007, 8(13):2135-47.
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