Dabigatran ethyl ester

CAS No. 429658-95-7

Dabigatran ethyl ester( Dabigatran ethyl ester | BIBR-951CL | BIBR 951CL | BIBR951CL | UNII-KJ4EH9410G )

Catalog No. M14458 CAS No. 429658-95-7

A reversible and selective, direct thrombin inhibitor (DTI) with Ki value of 4.5 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 32 In Stock
5MG 47 In Stock
10MG 86 In Stock
25MG 158 In Stock
50MG 270 In Stock
100MG 424 In Stock
200MG Get Quote In Stock
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Biological Information

  • Product Name
    Dabigatran ethyl ester
  • Note
    Research use only, not for human use.
  • Brief Description
    A reversible and selective, direct thrombin inhibitor (DTI) with Ki value of 4.5 nM.
  • Description
    A reversible and selective, direct thrombin inhibitor (DTI) with Ki value of 4.5 nM; an anticoagulant agent used to prevent stroke with atrial fibrillation.Thrombosis Approved.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    Dabigatran ethyl ester | BIBR-951CL | BIBR 951CL | BIBR951CL | UNII-KJ4EH9410G
  • Pathway
    Autophagy
  • Target
    Thrombin
  • Recptor
    Thrombin
  • Research Area
    Cardiovascular Disease
  • Indication
    Thrombosis

Chemical Information

  • CAS Number
    429658-95-7
  • Formula Weight
    499.5643
  • Molecular Formula
    C27H29N7O3
  • Purity
    >98% (HPLC)
  • Solubility
    10 mM in DMSO
  • SMILES
    O=C(OCC)CCN(C(C1=CC=C2C(N=C(CNC3=CC=C(C(N)=N)C=C3)N2C)=C1)=O)C4=NC=CC=C4
  • Chemical Name
    β-Alanine, N-[[2-[[[4-(aminoiminomethyl)phenyl]amino]methyl]-1-methyl-1H-benzimidazol-5-yl]carbonyl]-N-2-pyridinyl-, ethyl ester

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Wienen W, et al. Thromb Haemost. 2007 Jul;98(1):155-62. 2. Kansal AR, et al. Heart. 2012 Apr;98(7):573-8.
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