AG-14361

CAS No. 328543-09-5

AG-14361( AG14361 | AG-14361 | AG 14361. )

Catalog No. M14073 CAS No. 328543-09-5

AG14361 is a potent inhibitor of PARP1 with Ki of <5 nM. It is at least 1000-fold more potent than the benzamides.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 59 In Stock
5MG 128 In Stock
10MG 233 In Stock
25MG 453 In Stock
50MG 660 In Stock
100MG 888 In Stock
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Biological Information

  • Product Name
    AG-14361
  • Note
    Research use only, not for human use.
  • Brief Description
    AG14361 is a potent inhibitor of PARP1 with Ki of <5 nM. It is at least 1000-fold more potent than the benzamides.
  • Description
    AG14361 is a potent inhibitor of PARP1 with Ki of <5 nM. It is at least 1000-fold more potent than the benzamides.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    AG14361 | AG-14361 | AG 14361.
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    PARP
  • Recptor
    PARP1
  • Research Area
    Cancer
  • Indication
    ——

Chemical Information

  • CAS Number
    328543-09-5
  • Formula Weight
    320.39
  • Molecular Formula
    C19H20N4O
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: 12 mg/mL (37.45 mM)
  • SMILES
    O=C1C2=C3C(N=C(C4=CC=C(CN(C)C)C=C4)N3CCN1)=CC=C2
  • Chemical Name
    1-(4-((dimethylamino)methyl)phenyl)-8,9-dihydro-2,7,9a-triazabenzo[cd]azulen-6(7H)-one.

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Calabrese CR, et al. J Natl Y Inst, 2004, 96(1), 56-67.
molnova catalog
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