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AG-14361
CAS No. 328543-09-5
AG-14361( AG14361 | AG-14361 | AG 14361. )
Catalog No. M14073 CAS No. 328543-09-5
AG14361 is a potent inhibitor of PARP1 with Ki of <5 nM. It is at least 1000-fold more potent than the benzamides.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 121 | In Stock |
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| 2MG | 67 | In Stock |
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| 5MG | 110 | In Stock |
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| 10MG | 202 | In Stock |
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| 25MG | 394 | In Stock |
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| 50MG | 564 | In Stock |
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| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameAG-14361
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NoteResearch use only, not for human use.
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Brief DescriptionAG14361 is a potent inhibitor of PARP1 with Ki of <5 nM. It is at least 1000-fold more potent than the benzamides.
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DescriptionAG14361 is a potent inhibitor of PARP1 with Ki of <5 nM. It is at least 1000-fold more potent than the benzamides.
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In Vitro——
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In Vivo——
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SynonymsAG14361 | AG-14361 | AG 14361.
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PathwayCell Cycle/DNA Damage
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TargetPARP
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RecptorPARP1
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number328543-09-5
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Formula Weight320.39
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Molecular FormulaC19H20N4O
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Purity>98% (HPLC)
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SolubilityDMSO: 12 mg/mL (37.45 mM)
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SMILESO=C1C2=C3C(N=C(C4=CC=C(CN(C)C)C=C4)N3CCN1)=CC=C2
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Chemical Name1-(4-((dimethylamino)methyl)phenyl)-8,9-dihydro-2,7,9a-triazabenzo[cd]azulen-6(7H)-one.
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Calabrese CR, et al. J Natl Y Inst, 2004, 96(1), 56-67.
molnova catalog
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