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TG003
CAS No. 300801-52-9
TG003( —— )
Catalog No. M13931 CAS No. 300801-52-9
TG003 is a potent and ATP-competitive Cdc2-like kinase (Clk) inhibitor with IC50 of 20 nM, 200 nM, and 15 nM for Clk1, Clk2, and Clk4, respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 52 | In Stock |
|
| 5MG | 73 | In Stock |
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| 10MG | 126 | In Stock |
|
| 25MG | 251 | In Stock |
|
| 50MG | 429 | In Stock |
|
| 100MG | 628 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameTG003
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NoteResearch use only, not for human use.
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Brief DescriptionTG003 is a potent and ATP-competitive Cdc2-like kinase (Clk) inhibitor with IC50 of 20 nM, 200 nM, and 15 nM for Clk1, Clk2, and Clk4, respectively.
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DescriptionTG003 is a potent and ATP-competitive Cdc2-like kinase (Clk) inhibitor with IC50 of 20 nM, 200 nM, and 15 nM for Clk1, Clk2, and Clk4, respectively. No inhibitory effect on Clk3, SRPK1, SRPK2, or PKC.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayAngiogenesis
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TargetBcl-2
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RecptormCLK1| mCLK2| mCLK4
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Research Area——
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Indication——
Chemical Information
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CAS Number300801-52-9
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Formula Weight249.33
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Molecular FormulaC13H15NO2S
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Purity>98% (HPLC)
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SolubilityDMSO: 6 mg/mL warmed (24.06 mM)
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SMILESCCN\1C2=C(C=CC(=C2)OC)S/C1=C\C(=O)C
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Muraki M, et al. J Biol Chem. 2004, 279(23), 24246-24254.
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