Flopropione

CAS No. 2295-58-1

Flopropione( —— )

Catalog No. M13637 CAS No. 2295-58-1

Flopropione is a spasmolytic or antispasmodic agent, and acts as a 5-HT1A receptor antagonist.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 42 In Stock
50MG 28 In Stock
100MG 37 In Stock
200MG 52 In Stock
500MG 86 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Flopropione
  • Note
    Research use only, not for human use.
  • Brief Description
    Flopropione is a spasmolytic or antispasmodic agent, and acts as a 5-HT1A receptor antagonist.
  • Description
    Flopropione is a spasmolytic or antispasmodic agent, and acts as a 5-HT1A receptor antagonist(In Vivo):The effect of Flopropione as an antispasmodic agent on the rate of passing a calculus from the urinary tract has been compared retrospectively with patients in whom passage was spontaneous. Flopropine has been shown, with statistical significance, to be superior to the control in cumulative passage rate after initiation of administration. Flopropine has been shown to exert a spasmolytic effect not only on smooth muscle of the gastrointestinal tract but also on smooth muscle of the pancreatobiliary and urinary systems.
  • In Vitro
    ——
  • In Vivo
    The effect of Flopropione as an antispasmodic agent on the rate of passing a calculus from the urinary tract has been compared retrospectively with patients in whom passage was spontaneous. Flopropine has been shown, with statistical significance, to be superior to the control in cumulative passage rate after initiation of administration. Flopropine has been shown to exert a spasmolytic effect not only on smooth muscle of the gastrointestinal tract but also on smooth muscle of the pancreatobiliary and urinary systems.
  • Synonyms
    ——
  • Pathway
    Endocrinology/Hormones
  • Target
    5-HT Receptor
  • Recptor
    5-HT1A
  • Research Area
    Neurological Disease
  • Indication
    ——

Chemical Information

  • CAS Number
    2295-58-1
  • Formula Weight
    182.18
  • Molecular Formula
    C9H10O4
  • Purity
    >98% (HPLC)
  • Solubility
    Ethanol: 36 mg/mL (197.61 mM); DMSO: 36 mg/mL (197.61 mM)
  • SMILES
    CCC(=O)C1=C(O)C=C(O)C=C1O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Aso Y, et al. J Pharm Sci, 2000, 89(3), 408-416.
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