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Atagabalin
CAS No. 223445-75-8
Atagabalin( PD 0200390 )
Catalog No. M13581 CAS No. 223445-75-8
Atagabalin (PD 0200390) is a novel ligand of the voltage-dependent calcium channel (VDCC) α2δ subunit (1 and 2) for treatment for insomnia.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 873 | Get Quote |
|
| 50MG | 1782 | Get Quote |
|
| 100MG | 2250 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NameAtagabalin
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NoteResearch use only, not for human use.
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Brief DescriptionAtagabalin (PD 0200390) is a novel ligand of the voltage-dependent calcium channel (VDCC) α2δ subunit (1 and 2) for treatment for insomnia.
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DescriptionAtagabalin (PD 0200390) is a novel ligand of the voltage-dependent calcium channel (VDCC) α2δ subunit (1 and 2) for treatment for insomnia.Sleep Disorder Phase 2 Discontinued.
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In Vitro——
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In Vivo——
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SynonymsPD 0200390
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PathwayGPCR/G Protein
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TargetCalcium Channel
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RecptorCalcium Channel
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Research AreaNeurological Disease
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IndicationSleep Disorder
Chemical Information
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CAS Number223445-75-8
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Formula Weight185.267
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Molecular FormulaC10H19NO2
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Purity>98% (HPLC)
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Solubility——
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SMILESO=C(O)CC1(CN)C[C@H](C)[C@@H](C)C1
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Chemical Name2-((3S,4S)-1-(aminomethyl)-3,4-dimethylcyclopentyl)acetic acid
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Blakemore DC, et al. Bioorg Med Chem Lett. 2010 Jan 15;20(2):461-4.
2. Quintero JE, et al. Brain Res. 2011 Jul 15;1401:1-9.
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