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Atagabalin

CAS No. 223445-75-8

Atagabalin( PD 0200390 )

Catalog No. M13581 CAS No. 223445-75-8

Atagabalin (PD 0200390) is a novel ligand of the voltage-dependent calcium channel (VDCC) α2δ subunit (1 and 2) for treatment for insomnia.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    Atagabalin
  • Note
    Research use only, not for human use.
  • Brief Description
    Atagabalin (PD 0200390) is a novel ligand of the voltage-dependent calcium channel (VDCC) α2δ subunit (1 and 2) for treatment for insomnia.
  • Description
    Atagabalin (PD 0200390) is a novel ligand of the voltage-dependent calcium channel (VDCC) α2δ subunit (1 and 2) for treatment for insomnia.Sleep Disorder Phase 2 Discontinued.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    PD 0200390
  • Pathway
    GPCR/G Protein
  • Target
    Calcium Channel
  • Recptor
    Calcium Channel
  • Research Area
    Neurological Disease
  • Indication
    Sleep Disorder

Chemical Information

  • CAS Number
    223445-75-8
  • Formula Weight
    185.267
  • Molecular Formula
    C10H19NO2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    O=C(O)CC1(CN)C[C@H](C)[C@@H](C)C1
  • Chemical Name
    2-((3S,4S)-1-(aminomethyl)-3,4-dimethylcyclopentyl)acetic acid

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Blakemore DC, et al. Bioorg Med Chem Lett. 2010 Jan 15;20(2):461-4. 2. Quintero JE, et al. Brain Res. 2011 Jul 15;1401:1-9.
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