CAM4066

CAS No. 2101206-81-7

CAM4066( CAM 4066 | CAM-4066 )

Catalog No. M13331 CAS No. 2101206-81-7

CAM4066 (CAM-4066) is a potent and selective CK2α inhibitor with Kd of 0.32 uM and IC50 of 0.37 uM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    CAM4066
  • Note
    Research use only, not for human use.
  • Brief Description
    CAM4066 (CAM-4066) is a potent and selective CK2α inhibitor with Kd of 0.32 uM and IC50 of 0.37 uM.
  • Description
    CAM4066 (CAM-4066) is a potent and selective CK2α inhibitor with Kd of 0.32 uM and IC50 of 0.37 uM, shows significantly improved selectivity compared to other CK2α inhibitors.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    CAM 4066 | CAM-4066
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    Casein Kinase
  • Recptor
    Casein Kinase
  • Research Area
    Cancer
  • Indication
    ——

Chemical Information

  • CAS Number
    2101206-81-7
  • Formula Weight
    479.961
  • Molecular Formula
    C26H26ClN3O4
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    C1=CC=C(C=C1)C2=C(C=C(C=C2)CNCCC(=O)NCCC(=O)NC3=CC=CC(=C3)C(=O)O)Cl
  • Chemical Name
    3-(3-(3-(((2-chloro-[1,1'-biphenyl]-4-yl)methyl)amino)propanamido)propanamido)benzoic acid

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Iegre J, et al. Chem Sci. 2018 Feb 20;9(11):3041-3049. 2. Brear P, et al. Chem Sci. 2016 Nov 1;7(11):6839-6845. 3. De Fusco C, et al. Bioorg Med Chem. 2017 Jul 1;25(13):3471-3482.
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