Cart
sales@molnova.com
PDE6δ inhibitor 8
CAS No. 2088485-36-1
PDE6δ inhibitor 8( —— )
Catalog No. M13259 CAS No. 2088485-36-1
A novel selective small molecule inhibitor of PDE6δ/KRas interaction with Kd of 358 pM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 100MG | Get Quote | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
-
Product NamePDE6δ inhibitor 8
-
NoteResearch use only, not for human use.
-
Brief DescriptionA novel selective small molecule inhibitor of PDE6δ/KRas interaction with Kd of 358 pM.
-
DescriptionA novel selective small molecule inhibitor of PDE6δ/KRas interaction with Kd of 358 pM.
-
In Vitro——
-
In Vivo——
-
Synonyms——
-
PathwayMAPK/ERK Signaling
-
TargetRas
-
RecptorRas
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number2088485-36-1
-
Formula Weight675.256
-
Molecular FormulaC32H39ClN4O6S2
-
Purity>98% (HPLC)
-
Solubility——
-
SMILES——
-
Chemical Name2-amino-4-(((4-(N-(4-chlorobenzyl)-N-cyclopentylsulfamoyl)-N-(piperidin-4-ylmethyl)phenyl)sulfonamido)methyl)benzoic acid
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Martín-Gago P, et al. Angew Chem Int Ed Engl. 2017 Feb 20;56(9):2423-2428.
molnova catalog
related products
-
CMC2.24
CMC2.24 (TRB-N0224) is a novel tricarbonylmethane agent that inhibits the Ras-RAF-MEK-ERK pathway.
-
K-Ras G12C-IN-3
A novel and irreversible inhibitor of mutant K-ras G12C.
-
J-104871
J-104871 (UNII-6137X5QNJF) is a novel farnesyltransferase (FTase) inhibitor that competitively blocks Ras farnesylation in vivo, inhibits Ras processing in activated H-ras-transformed NIH3T3 cells, and suppresses tumor growth in nude mice transplanted with activated H-ras-transformed NIH3T3 cells.
