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Home - Products - GPCR/G Protein - Adrenergic Receptor - CL 316243

CL 316243

CAS No. 183720-02-7

CL 316243( BTA 243 )

Catalog No. M12836 CAS No. 183720-02-7

CL 316243 (BTA 243) is a potent, highly selective, orally active β3-adrenoceptor agonist with EC50 of 3 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    CL 316243
  • Note
    Research use only, not for human use.
  • Brief Description
    CL 316243 (BTA 243) is a potent, highly selective, orally active β3-adrenoceptor agonist with EC50 of 3 nM.
  • Description
    CL 316243 (BTA 243) is a potent, highly selective, orally active β3-adrenoceptor agonist with EC50 of 3 nM; Displays >10000-fold selective over β1 and β2 receptors; Significantly increases brown adipose tissue thermogenesis and resting metabolic rate in mice, also increases the concentration of insulin receptors and decreases the levels of serum insulin and blood glucose during the glucose overloading test.Obesity Discontinued.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    BTA 243
  • Pathway
    GPCR/G Protein
  • Target
    Adrenergic Receptor
  • Recptor
    Adrenergic Receptor
  • Research Area
    Metabolic Disease
  • Indication
    Obesity

Chemical Information

  • CAS Number
    183720-02-7
  • Formula Weight
    421.83
  • Molecular Formula
    C20H20ClNO7
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CC(CC1=CC2=C(C=C1)OC(O2)(C(=O)O)C(=O)O)NCC(C3=CC(=CC=C3)Cl)O
  • Chemical Name
    5-[(2R)-2-[[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino]propyl]-1,3-benzodioxole-2,2-dicarboxylic acid

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Berlan M, et al. J Pharmacol Exp Ther. 1994 Mar;268(3):1444-51. 2. Himms-Hagen J, et al. Am J Physiol. 1994 Apr;266(4 Pt 2):R1371-82. 3. Yoshida T, et al. Life Sci. 1994;54(7):491-8.
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