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BET bromodomain inhibitor
CAS No. 1505453-59-7
BET bromodomain inhibitor( MDK3597 | MDK-3597 | MDK 3597 | BET bromodomain inhibitor )
Catalog No. M12098 CAS No. 1505453-59-7
It is a BET bromodomain inhibitor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 76 | In Stock |
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| 2MG | 43 | In Stock |
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| 5MG | 69 | In Stock |
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| 10MG | 117 | In Stock |
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| 25MG | 198 | In Stock |
|
| 50MG | 272 | In Stock |
|
| 100MG | 431 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameBET bromodomain inhibitor
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NoteResearch use only, not for human use.
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Brief DescriptionIt is a BET bromodomain inhibitor.
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DescriptionIt is a BET bromodomain inhibitor.
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In Vitro——
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In Vivo——
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SynonymsMDK3597 | MDK-3597 | MDK 3597 | BET bromodomain inhibitor
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PathwayChromatin/Epigenetic
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TargetEpigenetic Reader Domain
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RecptorBET bromodomain
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Research Area——
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Indication——
Chemical Information
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CAS Number1505453-59-7
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Formula Weight400.26
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Molecular FormulaC20H15Cl2N3O2
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Purity>98% (HPLC)
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SolubilityDMSO: 10 mM
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SMILESO=C(N)C[C@@H]1N=C(C2=CC=C(Cl)C=C2)C3=CC(Cl)=CC=C3C4=C1ON=C4C
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Chemical Name(S)-2-[8-Chloro-6-(4-chloro-phenyl)-1-methyl-4H-3-oxa-2,5-diaza-benzo[e]azulen-4-yl]-acetamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Xiao Y, et al. Rheumatology (Oxford). 2015 Aug 3
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