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PU-WS13
CAS No. 1454619-14-7
PU-WS13( PU-WS-13 )
Catalog No. M11960 CAS No. 1454619-14-7
A potent and selective Grp94 inhibitor with Ic50 of 0.22 uM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 50MG | 659 | In Stock |
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| 100MG | Get Quote | In Stock |
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| 200MG | Get Quote | In Stock |
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| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NamePU-WS13
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NoteResearch use only, not for human use.
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Brief DescriptionA potent and selective Grp94 inhibitor with Ic50 of 0.22 uM.
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DescriptionA potent and selective Grp94 inhibitor with Ic50 of 0.22 uM; shows >35 fold selectivity over other four HSP90 paralogs, Hsp90α, Hsp90β and Trap-1 (IC50> 7 uM).
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In Vitro——
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In Vivo——
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SynonymsPU-WS-13
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PathwayCytoskeleton/Cell Adhesion Molecules
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TargetHSP
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RecptorHSP
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number1454619-14-7
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Formula Weight411.3519
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Molecular FormulaC17H20Cl2N6S
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Purity>98% (HPLC)
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SolubilityDMSO: ≥ 40 mg/mL
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SMILESNC1=C2N=C(SC3=CC(Cl)=CC(Cl)=C3)N(CCCNC(C)C)C2=NC=N1
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Chemical Name9H-Purine-9-propanamine, 6-amino-8-[(3,5-dichlorophenyl)thio]-N-(1-methylethyl)-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Patel PD, et al. Nat Chem Biol. 2013 Nov;9(11):677-84.
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