PD 123319 ditrifluoroacetate
CAS No. 136676-91-0
PD 123319 ditrifluoroacetate( PD123319 ditrifluoroacetate | PD-123319 ditrifluoroacetate )
Catalog No. M11516 CAS No. 136676-91-0
A potent, selective, non-peptide AT2 receptor with IC50 of 34 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 100MG | Get Quote | In Stock |
|
| 200MG | 896 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
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Biological Information
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Product NamePD 123319 ditrifluoroacetate
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NoteResearch use only, not for human use.
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Brief DescriptionA potent, selective, non-peptide AT2 receptor with IC50 of 34 nM.
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DescriptionA potent, selective, non-peptide AT2 receptor with IC50 of 34 nM.Heart Failure Discontinued.
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In Vitro——
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In Vivo——
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SynonymsPD123319 ditrifluoroacetate | PD-123319 ditrifluoroacetate
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PathwayGPCR/G Protein
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TargetAngiotensin Receptor
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RecptorAngiotensin Receptor
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Research AreaCardiovascular Disease
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Indication——
Chemical Information
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CAS Number136676-91-0
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Formula Weight736.6575
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Molecular FormulaC35H34F6N4O7
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Purity>98% (HPLC)
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SolubilityH2O: ≥ 36 mg/mL
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SMILESCC1=C(C=CC(=C1)CN2C=NC3=C2CC(N(C3)C(=O)C(C4=CC=CC=C4)C5=CC=CC=C5)C(=O)O)N(C)C.C(=O)(C(F)(F)F)O.C(=O)(C(F)(F)F)O
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Chemical Name1H-Imidazo[4,5-c]pyridine-6-carboxylic acid, 1-[[4-(dimethylamino)-3-methylphenyl]methyl]-5-(2,2-diphenylacetyl)-4,5,6,7-tetrahydro-, (6S)-, 2,2,2-trifluoroacetate (1:2)
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Blankley CJ, et al. J Med Chem. 1991 Nov;34(11):3248-60.
2. Keiser JA, et al. J Pharmacol Exp Ther. 1992 Sep;262(3):1154-60.
3. Macari D, et al. Eur J Pharmacol. 1993 Nov 2;249(1):85-93.
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