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RGFP 966
CAS No. 1357389-11-7
RGFP 966( RGFP966 | RGFP 966 | RGFP-966 )
Catalog No. M11466 CAS No. 1357389-11-7
RGFP966 is an HDAC3 inhibitor with IC50 of 0.08 μM in cell-free assay, exhibits > 200-fold selectivity over other HDAC.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 75 | In Stock |
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| 2MG | 42 | In Stock |
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| 5MG | 68 | In Stock |
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| 10MG | 107 | In Stock |
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| 25MG | 188 | In Stock |
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| 50MG | 291 | In Stock |
|
| 100MG | 477 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameRGFP 966
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NoteResearch use only, not for human use.
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Brief DescriptionRGFP966 is an HDAC3 inhibitor with IC50 of 0.08 μM in cell-free assay, exhibits > 200-fold selectivity over other HDAC.
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DescriptionRGFP966 is an HDAC3 inhibitor with IC50 of 0.08 μM in cell-free assay, exhibits > 200-fold selectivity over other HDAC.
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In Vitro——
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In Vivo——
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SynonymsRGFP966 | RGFP 966 | RGFP-966
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PathwayCell Cycle/DNA Damage
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TargetHDAC
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RecptorHDAC3
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number1357389-11-7
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Formula Weight362.4
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Molecular FormulaC21H19FN4O
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Purity>98% (HPLC)
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SolubilityDMSO: ≥100mM
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SMILESO=C(NC1=CC=C(F)C=C1N)/C=C/C2=CN(C/C=C/C3=CC=CC=C3)N=C2.
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Chemical Name(E)-N-(2-amino-4-fluorophenyl)-3-(1-cinnamyl-1H-pyrazol-4-yl)acrylamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Malvaez M, et al. PNAS, 2013, 110(7), 2647-2652.
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