Cart
sales@molnova.com
Neladenoson dalanate
CAS No. 1239309-58-0
Neladenoson dalanate( BAY 10-67197 )
Catalog No. M10962 CAS No. 1239309-58-0
Neladenoson dalanate is a potent, selective, orally acitve partial adenosine A1 receptor (A1AR) agonist (EC50=0.1 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 873 | Get Quote |
|
| 50MG | 1782 | Get Quote |
|
| 100MG | 2250 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
-
Product NameNeladenoson dalanate
-
NoteResearch use only, not for human use.
-
Brief DescriptionNeladenoson dalanate is a potent, selective, orally acitve partial adenosine A1 receptor (A1AR) agonist (EC50=0.1 nM).
-
DescriptionNeladenoson dalanate is a potent, selective, orally acitve partial adenosine A1 receptor (A1AR) agonist (EC50=0.1 nM) for the treatment of chronic heart failure.Heart Failure Phase 2 Clinical.
-
In Vitro——
-
In Vivo——
-
SynonymsBAY 10-67197
-
PathwayApoptosis
-
TargetAdenosine Receptor
-
RecptorAdenosine Receptor
-
Research AreaCancer
-
Indication——
Chemical Information
-
CAS Number1239309-58-0
-
Formula Weight716.27
-
Molecular FormulaC35H34ClN7O4S2
-
Purity>98% (HPLC)
-
Solubility——
-
SMILESCC(C(=O)NC(C)C(=O)OCCOC1=CC=C(C=C1)C2=C(C(=NC(=C2C#N)SCC3=CSC(=N3)C4=CC=C(C=C4)Cl)N5CCCC5)C#N)N
-
Chemical Name2-{4-[2-({[2-(4-chlorophenyl)-1,3-thiazol- 4-yl]methyl}sulfanyl)-3,5-dicyano-6-(pyrrolidin-1-yl)pyridin- 4-yl]phenoxy}ethyl L-alanyl-L-alaninate
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Meibom D, et al. ChemMedChem. 2017 May 22;12(10):728-737.
2. Voors AA, et al. J Clin Pharmacol. 2017 Apr;57(4):440-451.
molnova catalog
related products
-
1-Ethyl-6-aminouraci...
1-Ethyl-6-aminouracil is an intermediate in the synthesis of a series of new substituted Xanthines which have high affinity and selectivity for the human adenosine A2B receptors.
-
ST-1535
A potent, selective A2A adenosine receptor antagonist with Ki of 6.6 nM.
-
Theophylline-7-aceti...
Theophylline-7-acetic acid is a stimulant drug of the xanthine chemical class. It acts as an adenosine receptor antagonist.
