AMPK activator 991

CAS No. 1219739-95-3

AMPK activator 991( —— )

Catalog No. M10830 CAS No. 1219739-95-3

AMPK activator 991 is an allosteric AMPK activator.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    AMPK activator 991
  • Note
    Research use only, not for human use.
  • Brief Description
    AMPK activator 991 is an allosteric AMPK activator.
  • Description
    AMPK activator 991 is an allosteric AMPK activator, activates non-phosphorylated Thr172 AMPK in vitro binds to α1β1γ1 and α2β1γ1 with Kd of 0.13 and 0.17 uM, respectively.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    AMPK
  • Recptor
    AMPK
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1219739-95-3
  • Formula Weight
    431.876
  • Molecular Formula
    C24H18ClN3O3
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CC1=C(C=C(C=C1)OC2=NC3=C(N2)C=C(C(=C3)C4=CC5=C(C=C4)C=CN5C)Cl)C(=O)O
  • Chemical Name
    5-((5-chloro-6-(1-methyl-1H-indol-6-yl)-1H-benzo[d]imidazol-2-yl)oxy)-2-methylbenzoic acid

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Willows R, et al. Biochem J. 2017 Aug 22;474(17):3059-3073. 2. Ngoei KRW, et al. Cell Chem Biol. 2018 Jun 21;25(6):728-737.e9.
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