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MS0124
CAS No. 1197196-63-6
MS0124( MS 0124 )
Catalog No. M10701 CAS No. 1197196-63-6
MS-0124 is a potent and selective inhibitor of G9a-like Protein (GLP) lysine methyltransferase with IC50 of 13 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 123 | In Stock |
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| 5MG | 117 | In Stock |
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| 10MG | 196 | In Stock |
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| 25MG | 392 | In Stock |
|
| 50MG | 616 | In Stock |
|
| 100MG | 861 | In Stock |
|
| 200MG | 1144 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameMS0124
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NoteResearch use only, not for human use.
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Brief DescriptionMS-0124 is a potent and selective inhibitor of G9a-like Protein (GLP) lysine methyltransferase with IC50 of 13 nM.
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DescriptionMS-0124 is a potent and selective inhibitor of G9a-like Protein (GLP) lysine methyltransferase with IC50 of 13 nM, shows >30-fold selectivity for GLP over G9a and other methyltransferases.
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In Vitro——
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In Vivo——
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SynonymsMS 0124
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PathwayChromatin/Epigenetic
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TargetHMTase
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RecptorHMTase
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Research Area——
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Indication——
Chemical Information
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CAS Number1197196-63-6
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Formula Weight387.484
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Molecular FormulaC20H29N5O3
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Purity>98% (HPLC)
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Solubility——
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SMILESCOC1=CC2=NC(N3CCOCC3)=NC(NC4CCN(C)CC4)=C2C=C1OC
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Chemical Name6,7-Dimethoxy-N-(1-methylpiperidin-4-yl)-2-morpholinoquinazolin-4-amine
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Xiong Y, et al. J Med Chem. 2017 Mar 9;60(5):1876-1891.
molnova catalog
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