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AZD6088

CAS No. 1131451-40-5

AZD6088( AZD-6088 | AZD 6088 )

Catalog No. M10458 CAS No. 1131451-40-5

AZD6088 (AZD-6088) is a potent and selective, orally bioavailable partial agonist of the M1 muscarinic receptor, reduces heat hyperalgesia in SNL rats with an EC50 of 46.6 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    AZD6088
  • Note
    Research use only, not for human use.
  • Brief Description
    AZD6088 (AZD-6088) is a potent and selective, orally bioavailable partial agonist of the M1 muscarinic receptor, reduces heat hyperalgesia in SNL rats with an EC50 of 46.6 nM.
  • Description
    AZD6088 (AZD-6088) is a potent and selective, orally bioavailable partial agonist of the M1 muscarinic receptor, reduces heat hyperalgesia in SNL rats with an EC50 of 46.6 nM.Pain Discontinued.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    AZD-6088 | AZD 6088
  • Pathway
    GPCR/G Protein
  • Target
    mAChR
  • Recptor
    mAChR
  • Research Area
    Neurological Disease
  • Indication
    Pain

Chemical Information

  • CAS Number
    1131451-40-5
  • Formula Weight
    406.571
  • Molecular Formula
    C22H38N4O3
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CC(C)OC(=O)N1CCC(CC1)(C)N2CCC(CC2)N3C4CCCCC4NC3=O
  • Chemical Name
    isopropyl 4'-methyl-4-((7aS)-2-oxooctahydro-1H-benzo[d]imidazol-1-yl)-[1,4'-bipiperidine]-1'-carboxylate

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Viberg A, et al. AAPS J. 2012 Dec;14(4):657-63. doi: 10.1208/s12248-012-9380-3.
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