Loratadine
CAS No. 79794-75-5
Loratadine ( Loratidine;SCH-29851 )
Catalog No. M15987 CAS No. 79794-75-5
A tricyclic antihistamine that acts as a selective inverse agonist of peripheral histamine H1-receptors.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
500MG | 37 | In Stock |
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1G | Get Quote | In Stock |
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Biological Information
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Product NameLoratadine
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NoteResearch use only, not for human use.
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Brief DescriptionA tricyclic antihistamine that acts as a selective inverse agonist of peripheral histamine H1-receptors.
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DescriptionA tricyclic antihistamine that acts as a selective inverse agonist of peripheral histamine H1-receptors.Allergy Approved
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SynonymsLoratidine;SCH-29851
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PathwayGPCR/G Protein
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TargetHistamine Receptor
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RecptorB(0)AT2
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Research AreaInflammation/Immunology
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IndicationAllergy
Chemical Information
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CAS Number79794-75-5
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Formula Weight382.88
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Molecular FormulaC22H23ClN2O2
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Purity>98% (HPLC)
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Solubility10 mM in DMSO
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SMILESCCOC(=O)N1CCC(=C2C3=C(CCC4=C2N=CC=C4)C=C(C=C3)Cl)CC1
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Chemical Name1-Piperidinecarboxylic acid, 4-(8-chloro-5,6-dihydro-11H-benzo[5,6]cyclohepta[1,2-b]pyridin-11-ylidene)-, ethyl ester
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Devillier P, et al. Clin Pharmacokinet. 2008;47(4):217-30.
2. Barnett A, et al. Agents Actions. 1984 Jun;14(5-6):590-7.
3. Roman IJ, et al. Clin Rev Allergy. 1993 Spring;11(1):89-110.
2. Barnett A, et al. Agents Actions. 1984 Jun;14(5-6):590-7.
3. Roman IJ, et al. Clin Rev Allergy. 1993 Spring;11(1):89-110.
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