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LY3143921
CAS No. 1627696-53-0
LY3143921 ( LY-3143921;LY 3143921 )
Catalog No. M12416 CAS No. 1627696-53-0
LY3143921 (LY-3143921) is an orally available, potent, selective inhibitor of Cdc7 kinase inhibitor, inhibits CDC7/DBF4 I and pMCM2 (S53) with IC50 values of 3.3 nM and 290 nM, respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 88 | Get Quote |
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| 10MG | 129 | Get Quote |
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| 25MG | 217 | Get Quote |
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| 50MG | 329 | Get Quote |
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| 100MG | 503 | Get Quote |
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| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameLY3143921
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NoteResearch use only, not for human use.
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Brief DescriptionLY3143921 (LY-3143921) is an orally available, potent, selective inhibitor of Cdc7 kinase inhibitor, inhibits CDC7/DBF4 I and pMCM2 (S53) with IC50 values of 3.3 nM and 290 nM, respectively.
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DescriptionLY3143921 (LY-3143921) is an orally available, potent, selective inhibitor of Cdc7 kinase inhibitor, inhibits CDC7/DBF4 I and pMCM2 (S53) with IC50 values of 3.3 nM and 290 nM, respectively.Solid Tumors Phase 1 Clinical
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SynonymsLY-3143921;LY 3143921
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PathwayAngiogenesis
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TargetCDK
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RecptorCDK
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Research AreaCancer
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IndicationSolid Tumors
Chemical Information
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CAS Number1627696-53-0
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Formula Weight327.32
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Molecular FormulaC16H14FN5O2
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Purity>98% (HPLC)
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Solubility——
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SMILESCC1(C2=C(C=C(C=C2)C3=CNN=C3)C(=O)N1)C4=NC=NC=C4F.O
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Chemical Name(3R)-3-(5-Fluoro-4-pyrimidinyl)-2,3-dihydro-3-methyl-6-(1H-pyrazol-4-yl)-1H-isoindol-1-one hydrate
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
molnova catalog
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