LSP-249

CAS No. 1801253-04-2

LSP-249( —— )

Catalog No. M23814 CAS No. 1801253-04-2

LSP-249 is a plasma kallikrein inhibitor under the study for angioedema, with an EC50 less than 100 nM in cell.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 36 In Stock
5MG 58 In Stock
10MG 87 In Stock
25MG 177 In Stock
50MG 295 In Stock
100MG 484 In Stock
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Biological Information

  • Product Name
    LSP-249
  • Note
    Research use only, not for human use.
  • Brief Description
    LSP-249 is a plasma kallikrein inhibitor under the study for angioedema, with an EC50 less than 100 nM in cell.
  • Description
    LSP-249 is a plasma kallikrein inhibitor under the study for angioedema, with an EC50 less than 100 nM in cell.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    kallikrein
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1801253-04-2
  • Formula Weight
    431.92
  • Molecular Formula
    C24H22ClN5O
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:31.25 mg/mL?(69.45 mM;?ultrasonic and warming and heat to 60°C)
  • SMILES
    Cc1cc(N)nc(C)c1CNC(c1cc(Cc2ccc3ncc(Cl)cc3c2)ncc1)=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Andrew Mcdonald, et al. Therapeutic inhibitory compounds. Patent. WO2016011209A1.
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