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LGD-3303
CAS No. 917891-35-1
LGD-3303( LGD3303 )
Catalog No. M16590 CAS No. 917891-35-1
LGD-3303 is an orally available, brain-penetrant nonsteroidal selective androgen receptor modulator (SARM) that that shows little or no cross-reactivity with related nuclear receptors.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 59 | In Stock |
|
| 10MG | 88 | In Stock |
|
| 50MG | 284 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameLGD-3303
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NoteResearch use only, not for human use.
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Brief DescriptionLGD-3303 is an orally available, brain-penetrant nonsteroidal selective androgen receptor modulator (SARM) that that shows little or no cross-reactivity with related nuclear receptors.
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DescriptionLGD-3303 is an orally available, brain-penetrant nonsteroidal selective androgen receptor modulator (SARM) that that shows little or no cross-reactivity with related nuclear receptors; has potent activity on levator ani muscle but is a partial agonist on the preputial gland and ventral prostate in a castrated rat model of androgen deficiency; enhances male-directed sexual preference, proceptive behavior, and lordosis behavior in sexually experienced, but not sexually naive, female rats.
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In Vitro——
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In Vivo——
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SynonymsLGD3303
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PathwayEndocrinology/Hormones
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TargetAndrogen Receptor (AR)
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RecptorAndrogenReceptor
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Research Area——
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Indication——
Chemical Information
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CAS Number917891-35-1
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Formula Weight342.743
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Molecular FormulaC16H14ClF3N2O
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Purity>98% (HPLC)
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SolubilityDMSO: Soluble （ < 1 mg/ml refers to the product slightly soluble or insoluble )
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SMILESO=C1NC2=C(C3=C(N(CC(F)(F)F)C(CC)=C3C)C=C2)C(Cl)=C1
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Chemical Name9-Chloro-2-ethyl-1-methyl-3-(2,2,2-trifluoroethyl)-3H-pyrrolo(3,2-F)quinolin-7(6H)-one
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Vajda EG, et al. J Pharmacol Exp Ther. 2009 Feb;328(2):663-70.
2. Vajda EG, et al. J Bone Miner Res. 2009 Feb;24(2):231-40.
3. Kudwa AE, et al. Endocrinology. 2010 Jun;151(6):2659-68.
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