Cart
sales@molnova.com
LGD-3303
CAS No. 917891-35-1
LGD-3303( LGD3303 )
Catalog No. M16590 CAS No. 917891-35-1
LGD-3303 is an orally available, brain-penetrant nonsteroidal selective androgen receptor modulator (SARM) that that shows little or no cross-reactivity with related nuclear receptors.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 59 | In Stock |
|
| 10MG | 88 | In Stock |
|
| 50MG | 284 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product NameLGD-3303
-
NoteResearch use only, not for human use.
-
Brief DescriptionLGD-3303 is an orally available, brain-penetrant nonsteroidal selective androgen receptor modulator (SARM) that that shows little or no cross-reactivity with related nuclear receptors.
-
DescriptionLGD-3303 is an orally available, brain-penetrant nonsteroidal selective androgen receptor modulator (SARM) that that shows little or no cross-reactivity with related nuclear receptors; has potent activity on levator ani muscle but is a partial agonist on the preputial gland and ventral prostate in a castrated rat model of androgen deficiency; enhances male-directed sexual preference, proceptive behavior, and lordosis behavior in sexually experienced, but not sexually naive, female rats.
-
In Vitro——
-
In Vivo——
-
SynonymsLGD3303
-
PathwayEndocrinology/Hormones
-
TargetAndrogen Receptor (AR)
-
RecptorAndrogenReceptor
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number917891-35-1
-
Formula Weight342.743
-
Molecular FormulaC16H14ClF3N2O
-
Purity>98% (HPLC)
-
SolubilityDMSO: Soluble （ < 1 mg/ml refers to the product slightly soluble or insoluble )
-
SMILESO=C1NC2=C(C3=C(N(CC(F)(F)F)C(CC)=C3C)C=C2)C(Cl)=C1
-
Chemical Name9-Chloro-2-ethyl-1-methyl-3-(2,2,2-trifluoroethyl)-3H-pyrrolo(3,2-F)quinolin-7(6H)-one
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Vajda EG, et al. J Pharmacol Exp Ther. 2009 Feb;328(2):663-70.
2. Vajda EG, et al. J Bone Miner Res. 2009 Feb;24(2):231-40.
3. Kudwa AE, et al. Endocrinology. 2010 Jun;151(6):2659-68.
molnova catalog
related products
-
UT-155
UT-155 is a selective and potent antagonist of the androgen receptor (AR) (Ki: 267 nM for UT-155 binding to AR-LBD).
-
Dihydrotestosterone(...
Dihydrotestosterone is a potent androgenic metabolite of testosterone. It is an agonist of the androgen receptor.
-
BAY 1024767
BAY 1024767 (BAY1024767) is a higly potent antagonist of androgen receptor (AR) wild-type (IC50=46 nM) and mutant forms located in the AR ligand-binding domain (LBD).
