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LDK1229
CAS No. 1800285-55-5
LDK1229( LDK 1229 )
Catalog No. M12734 CAS No. 1800285-55-5
LDK1229 is a novel potent, selective cannabinoid CB1 receptor inverse agonist with Ki of 220 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NameLDK1229
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NoteResearch use only, not for human use.
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Brief DescriptionLDK1229 is a novel potent, selective cannabinoid CB1 receptor inverse agonist with Ki of 220 nM.
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DescriptionLDK1229 is a novel potent, selective cannabinoid CB1 receptor inverse agonist with Ki of 220 nM; exhibits 3-fold relative selectivity for the CB1 over CB2, exhibits efficacy comparable with SR141716A in antagonizing the basal G protein coupling activity of CB1; increases cell surface localization of CB1 and structurally distinct from the first-generation CB1 inverse agonists.
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In Vitro——
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In Vivo——
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SynonymsLDK 1229
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PathwayGPCR/G Protein
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TargetCannabinoid Receptor
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RecptorCannabinoid Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number1800285-55-5
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Formula Weight434.956
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Molecular FormulaC24H29ClF2N2O
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical Name(4-(Bis(4-fluorophenyl)methyl)piperazin-1-yl)(cyclohexyl)methanone hydrochloride
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Mahmoud MM, et al. Mol Pharmacol. 2015 Feb;87(2):197-206.
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