DBEQ

CAS No. 177355-84-9

DBEQ( N,N'-Dibenzylquinazoline-2,4-diamine | JRF 12 )

Catalog No. M12670 CAS No. 177355-84-9

DBeQ(JRF-12) is a selective, potent, reversible, and ATP-competitive p97 inhibitor with IC50 of 1.5 μM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 44 In Stock
2MG 29 In Stock
5MG 44 In Stock
10MG 78 In Stock
25MG 155 In Stock
50MG 272 In Stock
100MG 345 In Stock
200MG 510 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    DBEQ
  • Note
    Research use only, not for human use.
  • Brief Description
    DBeQ(JRF-12) is a selective, potent, reversible, and ATP-competitive p97 inhibitor with IC50 of 1.5 μM.
  • Description
    DBeQ(JRF-12) is a selective, potent, reversible, and ATP-competitive p97 inhibitor with IC50 of 1.5 μM.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    N,N'-Dibenzylquinazoline-2,4-diamine | JRF 12
  • Pathway
    Proteasome/Ubiquitin
  • Target
    p97
  • Recptor
    p97
  • Research Area
    Cancer
  • Indication
    ——

Chemical Information

  • CAS Number
    177355-84-9
  • Formula Weight
    340.42
  • Molecular Formula
    C22H20N4
  • Purity
    >98% (HPLC)
  • Solubility
    Ethanol: 5 mg/mL (14.68 mM); DMSO: 68 mg/mL (199.75 mM)
  • SMILES
    C12=CC=CC=C1N=C(NCC3=CC=CC=C3)N=C2NCC4=CC=CC=C4
  • Chemical Name
    N2,N4-dibenzylquinazoline-2,4-diamine

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Chou TF, et al. Proc Natl Acad Sci U S A, 2011, 108(12), 4834-4839.
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