L-765314
CAS No. 189349-50-6
L-765314( —— )
Catalog No. M23865 CAS No. 189349-50-6
L-765314 is a drug which acts as a potent and selective antagonist for the Alpha-1 adrenergic receptor subtype α1B.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
2MG | 51 | In Stock |
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5MG | 80 | In Stock |
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10MG | 132 | In Stock |
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25MG | 258 | In Stock |
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50MG | 410 | In Stock |
|
100MG | 605 | In Stock |
|
200MG | Get Quote | In Stock |
|
500MG | Get Quote | In Stock |
|
1G | Get Quote | In Stock |
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Biological Information
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Product NameL-765314
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NoteResearch use only, not for human use.
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Brief DescriptionL-765314 is a drug which acts as a potent and selective antagonist for the Alpha-1 adrenergic receptor subtype α1B.
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DescriptionL-765314 is a drug which acts as a potent and selective antagonist for the Alpha-1 adrenergic receptor subtype α1B. It has mainly been used to investigate the role of α1B receptors in the regulation of blood pressure.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayApoptosis
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TargetAdenosine Receptor
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Recptorα1B-adrenergic receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number189349-50-6
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Formula Weight522.6
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Molecular FormulaC27H34N6O5
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Purity>98% (HPLC)
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SolubilityDMSO : 50 mg/mL (95.68 mM; Need ultrasonic)
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SMILESO=C(N1[C@H](C(NC(C)(C)C)=O)CN(C2=NC(N)=C3C=C(OC)C(OC)=CC3=N2)CC1)OCC4=CC=CC=C4
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Patane MA, et al. 4-Amino-2-[4-[1-(benzyloxycarbonyl)-2(S)- [[(1,1-dimethylethyl)amino]carbonyl]-piperazinyl]-6, 7-dimethoxyquinazoline (L-765,314): a potent and selective alpha1b adrenergic receptor antagonist. J Med Chem. 1998 Apr 9;41(8):1205-8.
molnova catalog
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