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Home - Products - GPCR/G Protein - Neurokinin Receptor - L-732138

L-732138

CAS No. 148451-96-1

L-732138 ( —— )

Catalog No. M21568 CAS No. 148451-96-1

L-732138 is a potent and competitive antagonist of neurokinin-1 (NK-1) receptor(IC50 : 2.3 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    L-732138
  • Note
    Research use only not for human use.
  • Brief Description
    L-732138 is a potent and competitive antagonist of neurokinin-1 (NK-1) receptor(IC50 : 2.3 nM).
  • Description
    L-732138 is a potent and competitive antagonist of neurokinin-1 (NK-1) receptor(IC50 : 2.3 nM).
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    Neurokinin Receptor
  • Recptor
    NK-1
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    148451-96-1
  • Formula Weight
    472.38
  • Molecular Formula
    C22H18F6N2O3
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)OCc1cc(cc(c1)C(F)(F)F)C(F)(F)F
  • Chemical Name
    [35-Bis(trifluoromethyl)phenyl]methyl (2S)-2-acetamido-3-(1H-indol-3-yl)propanoate

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Mu?oz M et al. The NK-1 Receptor Antagonist L-732138 Induces Apoptosis and Counteracts Substance P-Related Mitogenesis in Human Melanoma Cell Lines. Cancers (Basel). 2010 Apr 20;2(2):611-23.
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