KUNG38

CAS No. 1887033-00-2

KUNG38( KUNG-38 | KUNG 38 )

Catalog No. M12953 CAS No. 1887033-00-2

A potent, selective Grp94 inhibitor with Kd of 0.44 uM; displays 19-fold selecticity over Hsp90α.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
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50MG 2322 Get Quote
100MG 3060 Get Quote
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Biological Information

  • Product Name
    KUNG38
  • Note
    Research use only, not for human use.
  • Brief Description
    A potent, selective Grp94 inhibitor with Kd of 0.44 uM; displays 19-fold selecticity over Hsp90α.
  • Description
    A potent, selective Grp94 inhibitor with Kd of 0.44 uM; displays 19-fold selecticity over Hsp90α; induces the degradation of integrin α2 in MDA-MB-231 cells.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    KUNG-38 | KUNG 38
  • Pathway
    Cytoskeleton/Cell Adhesion Molecules
  • Target
    HSP
  • Recptor
    HSP
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1887033-00-2
  • Formula Weight
    411.24
  • Molecular Formula
    C18H16Cl2N2O5
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    ClC1=CC=C(CN2C=CN=C2CCC3=C(C(OC)=O)C(O)=CC(O)=C3Cl)O1
  • Chemical Name
    Methyl 3-Chloro-2-(2-(1-((5-chlorofuran-2-yl)methyl)-1H-imidazol-2-yl)ethyl)-4,6-dihydroxybenzoate

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Crowley VM, et al. J Med Chem. 2016 Apr 14;59(7):3471-88.
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