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KCL-286
CAS No. 1952276-71-9
KCL-286( —— )
Catalog No. M37200 CAS No. 1952276-71-9
KCL-286 is an orally available and potent retinoic acid receptor beta agonist for the amelioration of spinal cord injury (SCI).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 123 | Get Quote |
|
| 5MG | 187 | Get Quote |
|
| 10MG | 302 | Get Quote |
|
| 25MG | 615 | Get Quote |
|
| 50MG | 984 | Get Quote |
|
| 100MG | 1305 | Get Quote |
|
| 200MG | 1755 | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameKCL-286
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NoteResearch use only, not for human use.
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Brief DescriptionKCL-286 is an orally available and potent retinoic acid receptor beta agonist for the amelioration of spinal cord injury (SCI).
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DescriptionAnticancer agent 168 is an orally active retinoic acid receptor (RAR/RXR) beta2 agonist with ameliorating effects on spinal cord injury (SCI).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMetabolic Enzyme/Protease
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TargetRetinoid Receptor
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RecptorRetinoid Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number1952276-71-9
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Formula Weight334.33
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Molecular FormulaC19H14N2O4
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Purity>98% (HPLC)
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Solubility——
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SMILESO=C(O)C=1C=CC(=CC1)C2=NOC(=N2)C=3OC=4C(C3)=C(C=CC4C)C
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Goncalves MB, et al. Phase 1 safety, tolerability, pharmacokinetics and pharmacodynamic results of KCL-286, a novel retinoic acid receptor-β agonist for treatment of spinal cord injury, in male healthy participants. Br J Clin Pharmacol. 2023 Jul 15..?
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