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KA2507
CAS No. 1636894-46-6
KA2507 ( —— )
Catalog No. M23733 CAS No. 1636894-46-6
KA2507 is a potent and selective HDAC6 inibitor with an IC50 of 2.5nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 177 | In Stock |
|
| 10MG | 285 | In Stock |
|
| 25MG | 482 | In Stock |
|
| 50MG | 695 | In Stock |
|
| 100MG | 972 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameKA2507
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NoteResearch use only, not for human use.
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Brief DescriptionKA2507 is a potent and selective HDAC6 inibitor with an IC50 of 2.5nM.
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DescriptionKA2507 is a potent and selective HDAC6 inibitor with an IC50 of 2.5nM.
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Synonyms——
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PathwayCell Cycle/DNA Damage
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TargetHDAC
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RecptorHDAC6; HDAC8
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Research Area——
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Indication——
Chemical Information
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CAS Number1636894-46-6
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Formula Weight322.3
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Molecular FormulaC16H14N6O2
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Purity>98% (HPLC)
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SolubilityDMSO : 60 mg/mL (186.15 mM; Need ultrasonic)
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SMILESO=C(NO)C1=CC=C(CN(C2=NC=CN=C2)C3=NC=CN=C3)C=C1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Apostolia M Tsimberidou, et al. Preclinical Development and First-in-Human Study of KA2507, a Selective and Potent Inhibitor of Histone Deacetylase 6, for Patients with Refractory Solid Tumors. Clin Cancer Res. 2021 May 4.
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