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Imagabalin

CAS No. 610300-07-7

Imagabalin( PD 0332334 | PD 332334 )

Catalog No. M15291 CAS No. 610300-07-7

Imagabalin (PD 0332334) is a novel ligand for the α2δ subunit of the voltage-dependent calcium channel (VDCC) with some selectivity for the α2δ1 subunit over α2δ2.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

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Biological Information

Product Name

Imagabalin
Note

Research use only, not for human use.
Brief Description

Imagabalin (PD 0332334) is a novel ligand for the α2δ subunit of the voltage-dependent calcium channel (VDCC) with some selectivity for the α2δ1 subunit over α2δ2.
Description

Imagabalin (PD 0332334) is a novel ligand for the α2δ subunit of the voltage-dependent calcium channel (VDCC) with some selectivity for the α2δ1 subunit over α2δ2; demonstrated preclinical efficacy of anxiolytic, analgesic, hypnotic, and anticonvulsant-like activity for the treatment of generalized anxiety disorder.Anxiety Phase 3 Discontinued.
In Vitro

——
In Vivo

——
Synonyms

PD 0332334 | PD 332334
Pathway

GPCR/G Protein
Target

Calcium Channel
Recptor

Calcium Channel
Research Area

Neurological Disease
Indication

Anxiety

Chemical Information

CAS Number

610300-07-7
Formula Weight

173.253
Molecular Formula

C9H19NO2
Purity

>98% (HPLC)
Solubility

——
SMILES

CCC[C@@H](C)C[C@H](N)CC(O)=O
Chemical Name

(3S,5R)-3-amino-5-methyloctanoic acid

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Quintero JE, et al. Brain Res. 2011 Jul 15;1401:1-9.

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