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Upacicalcet

CAS No. 1333218-50-0

Upacicalcet( —— )

Catalog No. M34460 CAS No. 1333218-50-0

Upacicalcet (AJT-240) is an intraventricular calcium mimetic, a SHPT available for human hemodialysis, that inhibits excessive parathyroid hormone (PTH) secretion by directly acting on parathyroid cell membrane calcium-sensitive receptors, thereby lowering blood levels of PTH.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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5MG 257 In Stock
10MG 380 In Stock
25MG 635 In Stock
50MG 883 In Stock
100MG 1200 In Stock
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500MG 2399 In Stock
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Biological Information

  • Product Name
    Upacicalcet
  • Note
    Research use only, not for human use.
  • Brief Description
    Upacicalcet (AJT-240) is an intraventricular calcium mimetic, a SHPT available for human hemodialysis, that inhibits excessive parathyroid hormone (PTH) secretion by directly acting on parathyroid cell membrane calcium-sensitive receptors, thereby lowering blood levels of PTH.
  • Description
    Upacicalcet is an intravenous calcimimetic agent. Upacicalcet suppresses excessive parathyroid hormone (PTH) secretion, thereby lowering blood PTH levels, by acting directly on parathyroid cell membrane calcium-sensing receptors. Upacicalcet can be used for researching the disease of secondary hyperparathyroidism (SHPT).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    Calcium Channel
  • Recptor
    Calcium Channel
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1333218-50-0
  • Formula Weight
    351.76
  • Molecular Formula
    C11H14ClN3O6S
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    N(C(NC[C@@H](C(O)=O)N)=O)C1=CC(S(=O)(=O)O)=CC(Cl)=C1C
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Hoy SM. Upacicalcet: First Approval. Drugs. 2021;81(13):1593-1596. ?
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